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Dysregulated Proline Metabolism Exacerbates Hepatocellular Carcinoma Metastasis via EPRS1-Mediated mRNA Translation - PubMed

5 hours ago
  • #hepatocellular carcinoma metastasis
  • #EPRS1 translation
  • #proline metabolism
  • Proline metabolism is enhanced in hepatocellular carcinoma (HCC) metastasis, shown by increased proline levels and related enzymes in patients and mice.
  • High proline levels promote HCC metastasis by binding to EPRS1 at residue Glu1123, selectively boosting translation of PIK3CA, AKT3, and ITGB1 mRNAs.
  • The EPRS1 inhibitor bersiporocin blocks proline binding, suppresses protein translation, and inhibits metastasis in patient-derived xenograft models.