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Targeting genomic instability in cancer - PubMed

5 hours ago
  • #Cancer Therapeutics
  • #DNA Damage Response
  • #Genomic Instability
  • Genomic instability is a key feature of cancer, resulting from failures in DNA maintenance systems that allow genetic changes driving cancer.
  • Targeting genomic instability has evolved from chemotherapy and radiation to PARP inhibitors for HR-deficient tumors, and now includes ADCs and radiopharmaceuticals.
  • Precision medicine strategies aim to optimize patient selection, develop combination therapies, and improve the therapeutic index.
  • Multiple authors have conflicts of interest, including employment, commercial interests, funding, and consultancy roles with various pharmaceutical and biotech companies.