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Platelet RIP2 Limits Dense Granule Release and Thrombosis via DOCK8-Cdc42 - PubMed

5 hours ago
  • #myocardial infarction
  • #platelet activation
  • #thrombosis
  • RIP2 deficiency enhances platelet dense granule secretion and increases platelet aggregation and adhesion.
  • RIP2 inhibitor WEHI-345 potentiates human platelet dense granule secretion and inhibits RIP2 phosphorylation.
  • Lower RIP2 expression is observed in platelets from patients with coronary artery disease and mice with atherosclerosis.
  • RIP2 deficiency worsens myocardial infarction and cardiac function in a mouse ischemia/reperfusion model.
  • A novel pathway p-RIP2-DOCK8-Cdc42 suppresses dense granule release downstream of GPIb and GPVI activation.