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Liquiritin attenuates IONI-induced trigeminal neuropathic pain via TLR4/MyD88-dependent modulation of microglial M1-like polarization - PubMed

6 hours ago
  • #Neuropathic Pain
  • #Microglial Polarization
  • #TLR4/MyD88 Signaling
  • Liquiritin, a flavonoid from licorice, reduces trigeminal neuropathic pain induced by infraorbital nerve injury (IONI) in mice.
  • The mechanism involves suppression of microglial M1-like polarization and down-regulation of TLR4/MyD88 signaling, leading to decreased inflammatory cytokines (IL-1β, TNF-mall α) and pain mediators (CGRP, TRPV1).
  • In vivo and in vitro studies confirm Liquiritin's effects on pain behaviors and molecular markers, supported by network pharmacology and molecular docking data.
  • Preliminary safety assessment shows no significant liver enzyme changes at therapeutic doses, though serum creatinine increased, warranting further long-term safety studies.