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PRMT5 inhibition impairs Fanconi Anemia pathway-mediated homologous recombination and enhances the antitumor efficacy of Temozolomide in glioblastoma - PubMed

5 hours ago
  • #temozolomide
  • #PRMT5
  • #glioblastoma
  • PRMT5 inhibition enhances the cytotoxic effect of temozolomide in glioma stem-like cells.
  • PRMT5 inhibition impairs the Fanconi anemia pathway-mediated homologous recombination repair, increasing DNA damage.
  • Combination therapy of PRMT5 inhibitor and temozolomide reduces tumor growth and improves survival in mouse models.