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Molecular hydrogen triggers TRPC4-TRPC4AP-dependent reversible calcium transients via extracellular influx - PubMed

3 days ago
  • #TRPC4-TRPC4AP Axis
  • #Molecular Hydrogen
  • #Calcium Signaling
  • Molecular hydrogen (H2) triggers reversible calcium transients via extracellular influx.
  • H2 acts as a gaseous messenger, selectively opening plasma-membrane Ca2+ channels without causing cytotoxic overload.
  • The study used real-time calcium imaging, CRISPR-Cas9 gene editing, and in vivo imaging in mice to monitor Ca2+ signals.
  • H2-induced Ca2+ transients enhance cell motility, as confirmed by live-cell imaging and wound-healing assays.
  • Protein-protein docking revealed a dual-arginine cluster in TRPC4's CIRB domain essential for H2-evoked Ca2+ influx.
  • Mutating arginine residues in TRPC4 abolishes the H2-induced Ca2+ response.
  • H2 triggers proton efflux and increases intracellular pH, modulating TRPC4-TRPC4AP binding forces.
  • Transcriptomic analysis shows H2 activates calcium-related channels and promotes cytoskeletal remodeling and cell migration.
  • The study identifies H2 as a novel gaseous signaling molecule regulating Ca2+ channels via the TRPC4-TRPC4AP axis.