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Fisetin targets multiple signaling pathways to suppress microglia-mediated neuroinflammation and cognitive decline in Alzheimer's disease - PubMed

5 hours ago
  • #Alzheimer's disease
  • #Neuroinflammation
  • #Fisetin
  • Fisetin improves cognitive performance in APP/PS1 mice and reduces amyloid pathology.
  • Fisetin inhibits pro-inflammatory activation in microglia and reduces mitochondrial ROS overproduction.
  • PI3K identified as a key signaling node in fisetin's regulation of microglial inflammatory responses.
  • Fisetin modulates the PI3K-Akt-NF-κB axis to limit NF-κB nuclear translocation and cytokine release.
  • Conditioned medium from fisetin-treated microglia alleviates neuronal damage and restores BDNF and PSD95 expression.
  • PI3K may act as a molecular target of fisetin, highlighting its therapeutic potential in Alzheimer's disease.