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Identification of novel bioactive constituents from traditional decoction of jiao-tai-Wan based on "co-decoction reaction" and comparative analysis with formula granules - PubMed

11 hours ago
  • #co-decoction reaction
  • #diabetes mellitus
  • #formula granules
  • Study investigates therapeutic equivalence between formula granules and traditional co-decoction using Jiao-Tai-Wan in diabetic mice.
  • Identifies 29 new co-decoction-related compounds using UPLC-QE-Orbitrap-MS.
  • Co-decoction showed the most pronounced reduction in fasting blood glucose, followed by mixed decoction and formula granules.
  • Different preparations distinctly modulated gut microbiota in db/db mice.
  • Strong binding confirmed between main constituents (e.g., berberine, cinnamic acid) and taste receptors (TAS2R46, TRPV1).
  • Findings suggest co-decoction reaction products may explain efficacy differences between formula granules and traditional decoctions.