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Effect of gamma irradiation as terminal sterilization technique on the stability of oligonucleotides - PubMed

5 days ago
  • #sterilization
  • #oligonucleotides
  • #gamma-irradiation
  • Study explores gamma irradiation for terminal sterilization of oligonucleotides.
  • Evaluated radioprotective factors: glycerine, histidine, trehalose, ascorbate, and dry ice.
  • Homo-oligomers of deoxythymidine (5-45-mers) used as representative oligonucleotides.
  • UPLC method with diode array detection quantified degradation accurately.
  • Best integrity observed in samples without stabilizers at 25 kGy (5.2%-13.2% degradation).
  • Histidine, trehalose, and ascorbate increased degradation (9.5%-24.2%).
  • Glycerin caused extensive degradation (78.8%-96.8%).
  • Dry ice during irradiation showed no protective benefit and slightly increased degradation.
  • Gamma irradiation works best for oligonucleotide sterilization in aqueous solution without radioprotective factors.