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Insulin increases expression of cannabinoid receptor 1 by suppressing lysosomal degradation via ERK signaling pathway - PubMed

4 hours ago
  • #insulin
  • #cannabinoid receptor 1
  • #ERK signaling
  • Insulin increases CB1R expression in hepatocytes by activating ERK signaling and inhibiting lysosomal degradation.
  • Inhibition of ERK blocks insulin-induced CB1R expression, indicating ERK pathway involvement.
  • Insulin suppresses lysosomal degradation of CB1R, stabilizing the receptor and enhancing its effects.
  • Hyperinsulinemia exacerbates MASLD/MASH via the insulin-ERK-CB1R axis, suggesting a potential therapeutic target.