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Polysaccharide-based inflammatory microenvironment-responsive nanocarriers for ulcerative colitis: Advances in design, mechanisms, and therapeutic applications - PubMed

5 hours ago
  • #ulcerative-colitis
  • #nanocarriers
  • #drug-delivery
  • Polysaccharide-based inflammatory microenvironment-responsive nanocarriers (PIMRNs) offer novel opportunities for ulcerative colitis (UC) management.
  • PIMRNs exhibit bioactivity, biocompatibility, and multifunctional modulation capabilities, enabling precise targeting and controlled drug release.
  • The inflammatory microenvironment of UC, including elevated reactive oxygen species, dysregulated pH, and enzyme overexpression, triggers PIMRNs for spatiotemporally controlled drug release.
  • PIMRNs enhance therapeutic efficacy while minimizing off-target adverse effects, potentially transforming UC treatment paradigms.
  • The review outlines recent advances in PIMRNs, design principles, optimization strategies, and challenges for clinical translation.