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Unraveling the potential of targeting methionine metabolism in cancer - PubMed

5 hours ago
  • #immunotherapy
  • #cancer
  • #methionine metabolism
  • Methionine metabolism is crucial for cellular homeostasis, affecting protein synthesis, redox regulation, and epigenetic control.
  • Cancer cells rely heavily on methionine, especially for S-adenosylmethionine (SAM) synthesis, which supports oncogenic transcriptional programs.
  • Methionine adenosyltransferase 2A (MAT2A), an enzyme involved in SAM production, is often overexpressed in tumors.
  • Dysregulated methionine metabolism impacts the tumor microenvironment (TME), affecting nutrient competition and antitumor immunity.
  • MAT2A is identified as a metabolic vulnerability in cancer, with potential for synthetic lethality-based targeting.
  • Methionine-restricted strategies and MAT2A inhibition are emerging as promising interventions that may enhance immunotherapy efficacy.
  • The review outlines the clinical potential of methionine-targeted therapies and future research directions in cancer treatment.