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KIF20A inhibits TRIM21-dependent ubiquitination of DHX9 to boost SOX2 stability, enhancing OSCC stemness and ferroptosis resistance - PubMed

3 months ago
  • #OSCC
  • #KIF20A
  • #ferroptosis
  • KIF20A is overexpressed in OSCC and linked to poor clinical outcomes.
  • KIF20A interacts with DHX9, inhibiting its TRIM21-mediated ubiquitination and degradation.
  • Stabilized DHX9 enhances SOX2 mRNA stability, promoting CSC maintenance and ferroptosis resistance.
  • KIF20A activates the PI3K/AKT pathway, supporting stemness and ferroptosis resistance in OSCC.
  • ENMD-2076 reduces KIF20A expression, attenuates CSC traits, and enhances cisplatin sensitivity.
  • Targeting KIF20A may improve therapeutic outcomes in OSCC, either alone or with chemotherapy.