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Antidiabetic drug effects on gastrointestinal health: convergent evidence from a longitudinal cohort and Mendelian randomization study - PubMed

19 hours ago
  • #Antidiabetic drugs
  • #Mendelian randomization
  • #Gastrointestinal health
  • Sulfonylurea use is associated with a lower risk of colorectal cancer (CRC) compared to non-sulfonylurea users (HR: 0.76).
  • Insulin use is linked to a decreased risk of diverticular disease versus non-insulin users (HR: 0.75).
  • Combination therapy of metformin with sulfonylureas further reduces CRC risk (HR: 0.61).
  • Post-metformin use of DPP-4 inhibitors with sulfonylureas or GLP-1 receptor agonists increases acute pancreatitis risk.
  • Mendelian randomization validates that sulfonylureas targeting INS reduce CRC risk (OR: 0.56) and insulin targeting LRP2 reduces diverticular disease risk (OR: 0.89).
  • Antidiabetic regimens, including combinations and sequences, are clinically important for preventing gastrointestinal morbidity in type 2 diabetes patients, highlighting the need for personalized treatment.