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PIEZO1 regulates smooth muscle cell plasticity by integrating mechanical stretch with glycolytic metabolism - PubMed

4 hours ago
  • #PIEZO1
  • #vascular remodeling
  • #glycolytic metabolism
  • PIEZO1 plays a critical role in pulmonary artery smooth muscle cell (PASMC) plasticity by integrating mechanical stretch with glycolytic metabolism.
  • Under hypoxia, PIEZO1 activation promotes glycolysis in PASMCs via HIF1α and PFKFB3, leading to lactate production and cell proliferation.
  • In severe pulmonary injury, hyper-activated PIEZO1 activates PPARγ, which antagonizes TGFβ signaling, restraining glycolysis and proliferation via FBP1.
  • Loss of smooth muscle Piezo1 attenuates hypoxia-induced PASMC growth and vascular remodeling but aggravates pulmonary fibrosis in mice.
  • The study identifies PIEZO1 as a key mediator of mechano-metabolic coupling in PASMCs during pulmonary vascular remodeling.