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Matrine improves bile acid metabolism and reduces inflammatory and oxidative stress in colitis via the JAK2 pathway - PubMed

4 hours ago
  • #JAK2 Pathway
  • #Colitis
  • #Bile Acid Metabolism
  • Matrine targets JAK2 directly, as shown by molecular docking.
  • In colitis models, matrine reduces inflammation by lowering cytokines like IL-1β, TNF-α, and IL-6.
  • Matrine decreases oxidative stress markers, including reactive oxygen species (ROS).
  • It restores bile acid homeostasis by upregulating transporters MRP3 and MRP4 and receptor FXR.
  • JAK2 overexpression reverses matrine's therapeutic effects, confirming JAK2-dependent mechanism.
  • Findings validated in human ulcerative colitis patients, showing relevance to clinical conditions.