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Ganoderic Acids Alleviate Neuroinflammation by Targeting Myeloid Differentiation Factor 2 for Ischemic Stroke Therapy - PubMed

a day ago
  • #ganoderic acid
  • #ischemic stroke
  • #neuroinflammation
  • Ganoderic acids (GAs) from Ganoderma lucidum show anti-inflammatory properties.
  • GAs alleviate cerebral ischemic injury and inhibit microglial overactivation in stroke models.
  • GA-K, a monomer in GAs, targets myeloid differentiation protein 2 (MD2), blocking TLR4 interaction.
  • MD2 overexpression in ischemia is mitigated by GAs, reducing neuroinflammation via MAPK/NF-κB pathways.
  • MD2-deficient mice show reduced microglial activation and neuroprotection, unaffected by GAs.
  • GA-K's modulation of microglia through MD2 presents a therapeutic target for stroke.