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Betulin inhibits inflammatory factors synthesis in osteoarthritis synovial fibroblasts by suppressing the PI3K, Akt, and mTOR pathways and activating miR-5006-5p - PubMed

6 hours ago
  • #Betulin
  • #Osteoarthritis
  • #Inflammation
  • Betulin, extracted from birch trees, inhibits inflammatory factors CHI3L1 and ICAM-1 in osteoarthritis synovial fibroblasts (OASFs).
  • Levels of CHI3L1 and ICAM-1 are higher in OA patients and ACLT-induced OA rats compared to healthy individuals.
  • Betulin works by suppressing the PI3K, Akt, and mTOR pathways and activating miR-5006-5p to reduce inflammation.
  • Molecular docking analysis predicts direct interaction between betulin and CHI3L1/ICAM-1, suggesting potential for OA management.