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Lianhe Xiaozhi ointment ameliorates metabolic dysfunction-associated steatotic liver disease via peroxisome proliferator-activated receptor alpha pathway activation - PubMed

a day ago
  • #PPARα Pathway
  • #Liver Disease
  • #Traditional Chinese Medicine
  • Lianhe Xiaozhi ointment (LXO) is derived from Huanglian Wendan decoction and has a national invention patent.
  • LXO is recognized for treating metabolic disorders, especially metabolic dysfunction-associated steatotic liver disease (MASLD).
  • Six key bioactive components in LXO contribute to its efficacy against MASLD.
  • LXO provides multiple therapeutic effects: weight gain control, improved glucose/lipid metabolism, reduced liver injury, and gut microbiota correction.
  • LXO activates the peroxisome proliferator-activated receptor alpha (PPARα) pathway, crucial for its lipid-lowering effects.
  • In vitro studies confirm that PPARα antagonist reduces LXO's lipid-lowering capacity.
  • LXO's therapeutic benefits for MASLD are partly due to PPARα pathway activation.