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Retinoblastoma: unveiling molecular pathogenesis and pioneering organoid-driven therapeutic innovations - PubMed

2 hours ago
  • #Retinoblastoma
  • #Precision medicine
  • #Organoid model
  • Retinoblastoma (RB) is the most common pediatric intraocular malignancy, driven by RB1 inactivation.
  • Clinical challenges include treatment toxicity, relapse, and resistance.
  • Traditional models fail to replicate human RB genetics or tumor heterogeneity, necessitating advanced in vitro platforms.
  • Retinal organoids from human pluripotent or patient-specific stem cells enable 3D modeling of the tumor microenvironment, drug screening, and mechanistic studies.
  • Key RB pathogenesis factors: RB1 loss, MYCN amplification, epigenetic dysregulation (e.g., METTL3-mediated m6A), and dysregulated pathways (PI3K/AKT/mTOR, Hedgehog).
  • CRISPR-engineered organoids identify cone precursors as tumor origins and validate therapies like CDK4/6 inhibitors and sunitinib.
  • Organoid limitations: high costs, variable success rates, incomplete immune/vascular mimicry, and limited scalability.
  • Future directions: integrate multiomics, refine vascularization via 3D bioprinting, and develop immunocompetent models.
  • Organoid technology has potential to advance personalized therapies and improve patient survival and quality of life.