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Zinc finger proteins (ZFPs) in health and disease - PubMed

4 hours ago
  • #Gene regulation
  • #Therapeutic targets
  • #Zinc finger proteins
  • Zinc finger proteins (ZFPs) are a superfamily of DNA and RNA-binding proteins that regulate gene expression and cellular homeostasis.
  • ZFPs play critical roles in various human diseases, including cancer, neurological disorders, and autoimmune diseases.
  • Dysregulated ZFP activity contributes to disease pathogenesis, with ischemic stroke as a key example.
  • ZFPs influence stroke risk factors like hypertension, hyperglycemia, and atherosclerosis, and post-ischemic injury cascades such as neuroinflammation and blood-brain barrier disruption.
  • Therapeutic strategies targeting ZFPs include small-molecule modulators, PROTACs, ZFN-based gene editing, and nanocarrier delivery systems.
  • High-throughput computational screening is being used to develop precision therapies targeting ZFPs.
  • The review provides a framework for future research on ZFPs as therapeutic targets in ischemic stroke and other diseases.