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Carrier-Free Nano-Proteolysis Targeting Chimeras Enable Selective Protein Degradation and Enhance Photoimmunometabolic Therapy against Lung Adenocarcinoma - PubMed

a day ago
  • #immunotherapy
  • #lung adenocarcinoma
  • #nanoparticles
  • Carrier-free nanoparticles (MNC NPs) developed to enhance immunotherapy efficacy in lung adenocarcinoma.
  • NPs integrate BRD4-targeting PROTAC, A2AR antagonist, and photosensitizer for synergistic therapy.
  • Targets BRD4 and A2AR to alleviate immune resistance and reverse immunosuppression.
  • Photosensitizer enables photodynamic therapy, promoting tumor ablation and immune activation.
  • In vivo studies show suppression of primary, distant, and metastatic tumors.
  • Nano-PROTACs combine protein degradation, immunometabolic reprogramming, and photodynamic immunotherapy.